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Prescription Dry Eye Medications

Anti-inflammatory and MGD-directed therapies used in dry eye disease

Dry Eye Disease: Prescription Drop Strategy

When artificial tears are not enough

Non-preserved artificial tears can dilute inflammatory mediators and provide short-term symptom relief, but they do not reliably address the underlying drivers of moderate to severe dry eye disease (DED). In many patients, DED behaves as a chronic, multifactorial inflammatory condition. Prescription therapy aims to reduce surface inflammation, stabilize the tear film, and support the lacrimal functional unit, in parallel with mechanical and environmental measures.

Start with the dominant mechanism

DED management is most effective when it is mechanism-based. Document whether signs and symptoms point primarily to aqueous deficiency, evaporative disease from meibomian gland dysfunction (MGD), or a mixed picture. Many patients have overlap, so treatment plans often combine an anti-inflammatory maintenance drop with targeted evaporative support, plus eyelid therapy and practical habit changes.

Immunomodulators for long-term control

Topical immunomodulators are a foundation for long-term pharmacologic management in aqueous-deficient or mixed DED. Their role is to down-regulate T-cell mediated inflammation affecting the lacrimal functional unit and ocular surface.

  • Cyclosporine A formulations: Calcineurin inhibitors (for example, cyclosporine 0.05% and 0.09%) reduce T-cell activation and cytokine release, with the goal of improving basal tear production and surface integrity over time. Clinical improvement is gradual, so counseling should set expectations that meaningful change may take several months of consistent twice-daily use.
  • Lifitegrast: An LFA-1 antagonist that interferes with T-cell adhesion and activation. Many patients report earlier symptom change than with traditional cyclosporine, sometimes within a few weeks, though sustained benefit still depends on regular ongoing dosing.

Choice between agents is guided by symptom profile, surface findings, prior response, tolerability, and formulary or coverage considerations. There is rarely a single best option for every patient.

Evaporative disease and MGD-focused therapy

In evaporative DED driven by MGD, improving the lipid layer is central. Lid hygiene, heat-based therapies, and in-office options are often paired with medications that reduce evaporation. Perfluorohexyloctane is a water-free drop designed to spread across the tear film and reduce evaporative loss. It is commonly positioned as an adjunct for patients with DED associated with MGD rather than a replacement for inflammation-directed maintenance therapy when inflammation or aqueous deficiency is also present.

Short-term steroid induction and flare control

Because immunomodulators act over weeks to months, many clinicians use a brief course of a soft topical steroid (for example, loteprednol or fluorometholone) as induction when starting long-term therapy or during symptomatic flares. A short taper can reduce surface inflammation, improve comfort, and enhance tolerance of the maintenance drop. As with any steroid, intraocular pressure monitoring and clear instructions about duration and taper matter.

Follow-up and realistic timelines

Prescription drops work best within a structured plan. Set expectations for timeline, document baseline signs, and schedule follow-up to reinforce adherence and adjust therapy. Treatment can be escalated or simplified as the ocular surface stabilizes, especially when eyelid therapy, environment, and systemic contributors are addressed in parallel.

Dry Eye Medications

BrandGenericDosingAmountAgesPregnancyMechanism
cyclosporine 0.09%bid60 vial box>18 yearsCimmunomodulator
loteprednol 0.25%qid (up to 14d)8.3mLNACester-based corticosteroid
perfluorohexyloctaneqid3mL>18 yearsNANA
Restasis
Generic
cyclosporine 0.05%bid30/60 vial tray5.5mL in 10mL bottle>16 yearsCimmunomodulator
acoltremon 0.003%bid60 vial cartonNANATRPM8 receptor agonist
varenicline 0.03mgbid4.2mL sprayNANAnicotinic acetylcholine agonistα-7 agonist
cyclosporine 0.1%bid2mL>18 yearsNAimmunomodulator
lifitegrast 5%bid60 vial carton>17 yearsNALFA-1 antagonist

Dry Eye Medication FAQs

How long does it take for cyclosporine or lifitegrast to work?

These medications are designed for long-term control rather than immediate relief. Some patients on lifitegrast notice symptom change within a few weeks, but a fair trial often requires 6 to 12 weeks. Cyclosporine formulations typically require several months of consistent twice-daily use before maximal benefit is evident. Setting expectations up front reduces early discontinuation and helps patients understand why supportive measures (non-preserved tears, lid therapy, and environmental adjustments) still matter during the ramp-up period.

Why do prescription dry eye drops sometimes burn on instillation?

Transient burning or stinging is common early on, especially when the ocular surface epithelium is inflamed or compromised. Some patients also notice taste disturbance or irritation as medication drains through the nasolacrimal system. Symptoms often improve as inflammation is controlled and the surface becomes healthier. Practical tips include using a non-preserved tear a few minutes before the prescription drop, spacing products appropriately, and reviewing instillation technique.

Can perfluorohexyloctane (MGD-focused drops) be used with contact lenses?

Most product labeling advises not instilling perfluorohexyloctane while contact lenses are in place. Patients should remove lenses before use and follow the specific product instructions for when lenses can be reinserted. For contact lens wearers with DED or MGD, it often helps to pair medication with a lens strategy that reduces surface stress, such as daily disposable lenses or reduced wear time, based on the overall plan.

Why use a short steroid when starting long-term dry eye therapy?

Immunomodulators typically take weeks to months to reduce inflammation. A short course of a soft topical steroid is sometimes used at the start or during a flare to calm surface inflammation more quickly, improve comfort, and make long-term drops easier to tolerate. Steroids require clear stop and taper instructions and appropriate intraocular pressure monitoring.